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Cardiovascular Dilated cardiomyopathy disease

TYA-018 is an Orally Active HDAC6 Inhibitor for Cardiovascular Disease Research

Edward Jenner 2023-05-26

Dilated cardiomyopathy (DCM) is a form of heart muscle weakness. Firstly, it shows the reduction of cardiac output, as well as thinning and enlargement of left ventricular chambers. Secondly, DCM…

Malaria

FNDR-20123 is an Orally Active and a First-in-Class Anti-Malarial HDAC Inhibitor

Edward Jenner 2021-03-20

Malaria remains one of the most severe and life-threatening infectious diseases. Among the various Plasmodium spp., Plasmodium falciparum is the most virulent and life-threatening form, prevailing in Southeast Asia and Africa.…

HIV Viral Immunology

BRD3308, a Highly Selective HDAC3 Inhibitor, Activates HIV-1 Transcription and Disrupts HIV-1 Latency

Edward Jenner 2020-05-02

Histone deacetylases (HDAC) are a class of enzymes that remove acetyl groups from an ε-N-acetyl-lysine amino acid on a histone. Specifically, selective HDAC inhibitors are as a potential anti latent…

Cancer Immunology

Pivanex is an Orally Active HDAC Inhibitor with Antimetastic and Antiangiogenic Properties

Edward Jenner 2020-04-11

Many malignancies, particularly leukemias, are associated with aberrant recruitment of histone deacetylases (HDACs) or with mutations in histone acetyltransferases such as EP300. In addition, Histone acetylation plays a key role…

Fibrosis Renal Fibrosis

CG-200745 Possesses Renoprotective Activity by Suppressing Renal Fibrosis and Inflammation

Edward Jenner 2019-10-18

In cancer, CG-200745 is a novel and potent hydroxamate-based pan-HDAC inhibitor. Moreover, another study from Hong Sang Choi demonstrated that CG200745 attenuates renal fibrosis in obstructive kidney disease. Epigenetic modifications…

HIV Viral Immunology

BRD-6929, a Selective HDAC 1/2 Inhibitor, Potentiates the Efficacy of GM Against Latent HIV-1

Edward Jenner 2019-09-10

Histone deacetylase (HDAC) enzymes, including subtypes comprising class I (HDAC1, HDAC2, HDAC3, and HDAC8) and class II (HDAC 4–7, HDAC9 and HDAC10), control the deacetylation of histone and non-histone proteins.…

Cancer Immunology Inflammation

FT895 is a Potent and Selective HDAC11 Inhibitor

Edward Jenner 2019-05-09

Histone deacetylases (HDACs) control protein acetylation levels. HDACs catalyze the removal of acetyl groups that are responsible for the addition of acetyl groups. The 11 HDAC family members require zinc…

Recent Posts

  • PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH
  • Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research
  • Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research
  • Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research
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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

Immune System Research

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