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Tag: HIV

Cobicistat is a Selective CYP3A Inhibitor and a Pharmacokinetic Enhancer of HIV Inhibitors

2020-12-22 Edward Jenner

The highly active antiretroviral therapy (HAART) can transform the human immunodeficiency virus (HIV) infection into a manageable chronic disease in…

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Posted in: HIV, Viral Immunology Filed under: Antiviral, CYP3A, HIV

BRD3308, a Highly Selective HDAC3 Inhibitor, Activates HIV-1 Transcription and Disrupts HIV-1 Latency

2020-05-02 Edward Jenner

Histone deacetylases (HDAC) are a class of enzymes that remove acetyl groups from an ε-N-acetyl-lysine amino acid on a histone.…

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Posted in: HIV, Viral Immunology Filed under: Apoptosis, HDAC, HIV, Hyperglycaemia, Insulin, T Cell

PF-3450074 is a HIV-1 Capsid Protein Inhibitor

2020-03-24 Edward Jenner

Human immunodeficiency virus type 1 (HIV-1) infection leads to depletion of the immune dysfunction. Thereby results in immunodeficiency and vulnerability…

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Posted in: HIV, Viral Immunology Filed under: Antiviral, Capsid, HIV

ZL0580, a Selective BD1 BRD4 Inhibitor, Induces HIV Epigenetic Suppression

2020-03-12 Edward Jenner

HIV integrates its provirus into the host genome and establishes latent infection. Antiretroviral therapy (ART) can effectively suppress active HIV…

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Posted in: AIDs, HIV, Viral Immunology Filed under: BRD4, HIV, TAt

MS417 is a BET-Specific BRD4 Inhibitor

2020-01-17 Edward Jenner

NF-κB-mediated inflammation is a major pathology in kidney diseases, such as non-kidney inflammatory diseases, and rheumatoid arthritis. HIV infection in…

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Posted in: HIV, Inflammation, Rheumatoid Arthritis, Viral Immunology Filed under: BRD4, HIV, HIVAN, NF-κB

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