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Immune System Research
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Tag: ROS

Setanaxib (GKT137831) is an Orally Active And Specific NOX1/4 Inhibitor for Cardiovascular Disease Research

2023-05-16 Edward Jenner

NOX1 and NOX4 are two members of the NADPH oxidase family, as well as multiple transmembrane proteins on the cell…

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Posted in: Cardiovascular Filed under: MDA, NADPH Oxidase, ROS, Setanaxib

Praelolide is a Potent Nrf2 Activator, Suppresses Osteoclastogenesis and ROS Production

2023-01-03 Edward Jenner

Nrf2 is a transcription factor, that regulates the expression of antioxidant proteins. Besides, Nrf2 protects against oxidative damage triggered by…

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Posted in: Osteoarthritis Filed under: Nrf2, Osteoclastogenesis, Praelolide, ROS

Virodhamine, an Endocannabinoid, Regulates Neurotransmission

2022-12-02 Edward Jenner

The endogenous cannabinoid system consists of endogenous cannabinoids, cannabinoid receptors, and enzymes that synthesize and degrade endogenous cannabinoids. Specifically, many…

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Posted in: Alzheimer, Neurological Disease, Parkinson’s Filed under: cannabinoid receptor, CB1, CB2, endocannabinoid, ROS

OXSI-2 is an Oxindole Syk Inhibitor

2022-02-25 Edward Jenner

Spleen tyrosine kinase (Syk) is a 72 kDa non-receptor tyrosine kinase. Specifically, Syk is activated by binding the tandem SH2…

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Posted in: Inflammation Filed under: Caspase, IL-1β, Inflammasome, Pyroptosis, ROS

Blebbistatin is a Selective Non-Muscle Myosin II (NMII) Inhibitor

2022-02-16 Edward Jenner

Blebbistatin is a selective non-muscle myosin II (NMII) inhibitor, promotes directional migration of corneal endothelial cells (CECs) and accelerates wound healing,…

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Posted in: Inflammation, Metabolic Disorder Filed under: Corneal Edema, Myosin, NMII, ROS, Wound Healing

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