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Tag: Anti-Fibrotic

SC-236 is an Orally Active COX-2 Specific Inhibitor

2020-11-24 Edward Jenner

Liver fibrosis is the accumulation of connective tissue in the liver. The consequence results from an imbalance between production and…

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Posted in: Fibrosis, Inflammation Filed under: ALSS, Anti-Fibrotic, COX-2, NSAID, PPAR

KIRA-7 is an Allosteric IRE1α Kinase/Rnase Inhibitor

2020-02-25 Edward Jenner

Idiopathic pulmonary fibrosis (IPF) is a disease of progressive fibrosis and respiratory failure. Endoplasmic reticulum stress (ER stress) implicates in…

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Posted in: Fibrosis, Pulmonary Fibrosis Filed under: Anti-Fibrotic, ER Stress, IPF, IRE1α, Rnase

VU6015929 is a Selective and Orally Active Dual DDR1/2 Inhibitor

2020-01-19 Edward Jenner

Receptor tyrosine kinases are a large family of cell surface receptors responsible for regulating cellular proliferation, differentiation, survival, metabolism, and…

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Posted in: Pulmonary Fibrosis Filed under: Anti-Fibrotic, DDR, DMPK

FT011 is an Orally Active Anti-Fibrotic Agent

2019-08-26 Edward Jenner

Nowadays, fibrosis has become very familiar to us. It has different types based on the place where it occurs. Skin…

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Posted in: Chronic Heart Failure, Fibrosis, Inflammation Filed under: Anti-Fibrotic, Anti-Inflammatory, CHF
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