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Immune System Research
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Tag: Integrin

EMD527040 is a Highly Selective αvβ6 Antagonist with Antifibrotic Activities

2021-07-14 Edward Jenner

Integrin αvβ6 is a member of the arginyl glycyl aspartate (RGD) subfamily of heterodimer transmembrane glycoprotein receptor 9. Specifically, αvβ6…

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Posted in: Cancer Immunology, Fibrosis Filed under: Integrin, TGFβ, αvβ6

Lifitegrast (SAR 1118) is an Integrin LFA-1 (αLβ2) Antagonist

2021-07-05 Edward Jenner

Lymphocyte function-associated antigen 1 (LFA-1; αLβ2) is a key T cell integrin, which plays an important role in regulating T…

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Posted in: Inflammation Filed under: Diabete, ICAM-1, Integrin, LFA-1, αLβ2

THI0019 is a Potent Integrin α4β1 (VLA-4) Agonis

2020-11-14 Edward Jenner

Integrin α4β1 (VLA-4) promotes the immune system\’s inflammatory response by helping white blood cells move to tissues that need inflammation.…

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Posted in: Immunology Filed under: Integrin, Jurkat, SDF-1α, α4β1, α5β1, αLβ2

Firategrast is an Orally Bioavailable α4β1/α4β7 Integrin Antagonist

2020-11-11 Edward Jenner

Integrin α4β1 is an integrin dimer and is composed of CD49d (alpha 4) and CD29 (beta 1). Specifically, integrin α4β1 promotes the inflammatory response…

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Posted in: Multiple Sclerosis Filed under: Integrin, α4β1, α4β7

Leukadherin-1 is a Specific Agonist of the Leukocyte Surface αMβ2 Integrin CD11b/CD18

2020-11-05 Edward Jenner

In molecular biology, CD18 (integrin beta chain 2) is an integrin beta chain protein encoded by the human itgb2 gene.…

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Posted in: Inflammation, Lung Inflammation Filed under: CD11b, CD18, CR3, Integrin, αMβ2

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