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Tag: MAPK

IAXO-102, a TLR4 Antagonist, Inhibits Aortic Aneurysms Development

2019-09-06 Edward Jenner

Abdominal aortic aneurysm (AAA) is a localized enlargement of the abdominal aorta, larger than normal. It commonly causes no symptoms,…

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Posted in: Abdominal Aortic Aneurysm Filed under: MAPK, p65, TLR

LUT014, a B-Raf Inhibitor, Overrides MAP Kinase Pathway Inhibition in Healthy Epithelial Cells

2019-06-02 Edward Jenner

EGFR (Epidermal Growth Factor Receptor) is a receptor on the surface of cells which is expressed in many normal epithelial…

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Posted in: Skin Inflammation Filed under: B-Raf, MAPK

SB 203580, a Selective p38 MAPK Inhibitor, Inhibits Inflammatory Cytokine Production

2019-05-20 Edward Jenner

SB 203580 was identified as a selective p38 MAPK (p38 mitogen-activated protein kinases) inhibitor over 20 years ago. And it…

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Posted in: Inflammation Filed under: HSP, MAPK

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Anti-Inflammatory Anti-Tumor Antibacterial Antimalarial Antitumor Antiviral Apoptosis Autophagy Breast Cancer Btk Chemokines COPD COVID-19 COX Cytokine EGFR HBV HCV HDAC HIV IFN IL-6 IL-17 Infection Integrin Interferon Interleukin Leukemia Low Toxicity Multidrug Resistance Necroptosis NF-κB p38 MAPK PI3K PPI Proteasome RIPK STAT STING T Cell Th17 TLR TNF TNF-α α4β1
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