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Tag: NLRP3

GDC-2394 is an Orally Active and Selective NLRP3 Inhibitor

2022-11-24 Edward Jenner

Nucleotide oligomerization domain (NOD)-like receptors (NLRs) are critical cytoplasmic pattern-recognition receptors (PRRs) that play an important role in the host’s…

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Posted in: Immunology, Innate Immune Filed under: Anti-inflammatory Effect, IL-18, IL-1β, NLRP3

AMS-17 is a Potent NLRP3 Inhibitor, Inhibiting Microglia Activation

2022-07-07 Edward Jenner

Microglia is a kind of resident immune cell in the central nervous system (CNS) parenchyma. microglia remain in a quiescent…

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Posted in: Alzheimer, Neuroimmunology, Neurological Disease, Parkinson’s Filed under: brain injury, CNS disease, microglial clearance, N9 cell, neuro-inflammatory disease, neurological disorders, NLRP3

SCH-23390 is a Selective Dopamine D1-Like Receptor Antagonist

2021-12-28 Edward Jenner

Dopamine Receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Abnormal…

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Posted in: Neurological Disease Filed under: 5-HT, Dopamine, GIRK, Inflammasome, NLRP3, Potassium Channel

MCC7840 is a Potent and Selective Inhibitor of NLRP3 Inflammasome

2021-03-11 Edward Jenner

Inflammasomes are protein complexes that are important in several inflammatory diseases. Inflammasomes form part of the innate immune system that…

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Posted in: Inflammation Filed under: Inflammasome, NLRP3

Ac-FLTD-CMK, a GSDMD-Derived Inhibitor, is a Caspase Inhibitor

2020-12-05 Edward Jenner

Caspase is a family of protease that plays an important role in programmed cell death. Specifically, caspase also has other…

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Posted in: Inflammation Filed under: Apoptosis, Caspase, GSDMD, Inflammasome, NLRP3

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