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Tag: Low Toxicity

PACMA 31 is an Irreversible and Orally Active Protein Disulfide Isomerase (PDI) Inhibitor

2020-12-08 Edward Jenner

Ovarian cancer is one of the leading causes of death in women with gynecological cancers in the United States. About…

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Posted in: Cancer Immunology Filed under: ER Stress, Low Toxicity, Ovarian Cancer, PDI

UC-514321 Directly Targets STAT3/5 and Represses TET1 Expression Selectively

2020-03-17 Edward Jenner

Acute myeloid leukemia (AML) is a fatal form of hematopoietic malignancies. current treatment for AML involves multiple cycles of high-dose…

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Posted in: Cancer Immunology Filed under: Apoptosis, Low Toxicity, STAT, TET1

ML401 is a Selective EBI2/GPR183 Antagonist with Low Toxicity

2019-09-22 Edward Jenner

A robust antibody response is essential for efficient identification and eradication of pathogenic microbes and toxins. Dysregulation of the antibody…

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Posted in: Immunology Filed under: EBI2, GPR183, Low Toxicity

Evobrutinib is an Orally Active BTK Inhibitor for Immunological Diseases Treatment

2019-08-15 Edward Jenner

Bruton’s tyrosine kinase (BTK), a member of the Tec family of tyrosine kinases, is expressed in B cells, macrophages, and…

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Posted in: Autoimmune Disorders, Rheumatoid Arthritis, Systemic Lupus Erythematosus Filed under: Anti-Inflammatory, Btk, Low Toxicity

AZD7624 Is an Inhaled p38 Inhibitor with Minimal Systemic Exposure

2019-07-27 Edward Jenner

Chronic obstructive pulmonary disease (COPD) is a kind of lung disease. The symptoms are obvious, including shortness of breath and…

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Posted in: Inflammation Filed under: Anti-Inflammatory, Low Toxicity, p38

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Anti-Inflammatory Anti-Tumor Antibacterial Antimalarial Antitumor Antiviral Apoptosis Autophagy Breast Cancer Btk Chemokines COPD COX Cytokine EGFR ER Stress HBV HCV HDAC HIV IFN IL-6 IL-17 Infection Integrin Interferon Interleukin Leukemia Low Toxicity Multidrug Resistance Necroptosis NF-κB p38 MAPK PI3K PPI Proteasome RIPK STAT STING T Cell Th17 TLR TNF TNF-α α4β1
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