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Tag: Low Toxicity

KL1333, a β-lapachone Derivative , is an Orally Available NAD+ Modulator

2022-01-22 Edward Jenner

Mitochondria is an essential organelle, and it generates most of the energy required by the human body in the form…

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Posted in: Metabolic Disease Filed under: AMPK, Low Toxicity, NAD, Ototoxicity, PGC-1α, SIRT1

FV-100 is a Selective and Orally Active Anti-Varicella Zoster Virus Agent

2021-07-16 Edward Jenner

Varicella zoster virus (VZV) is a double-stranded DNA alphaherpesvirus. And it is associated with seasonal outbreaks of varicella in nonimmunized…

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Posted in: Viral Immunology Filed under: Low Toxicity, Zoster

ACH-000143 is an Orally Active Melatonin Receptor Agonist

2021-05-17 Edward Jenner

The melatonin receptor is a G protein-coupled receptor (GPCR) that binds to melatonin. Specifically, receptors are crucial in the signal cascade…

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Posted in: Metabolic Disease Filed under: Low Toxicity, Melatonin, Obese, Plasma Glucose, Weight Control

PACMA 31 is an Irreversible and Orally Active Protein Disulfide Isomerase (PDI) Inhibitor

2020-12-08 Edward Jenner

Ovarian cancer is one of the leading causes of death in women with gynecological cancers in the United States. About…

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Posted in: Cancer Immunology Filed under: ER Stress, Low Toxicity, Ovarian Cancer, PDI

UC-514321 Directly Targets STAT3/5 and Represses TET1 Expression Selectively

2020-03-17 Edward Jenner

Acute myeloid leukemia (AML) is a fatal form of hematopoietic malignancies. current treatment for AML involves multiple cycles of high-dose…

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Posted in: Cancer Immunology Filed under: Apoptosis, Low Toxicity, STAT, TET1

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