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Tag: Antibacterial

BPH-1358 is a Dual FPPS and UPPS Inhibitor

2019-11-11 Edward Jenner

As we all know, Farnesyl diphosphate synthase(FPPS) is an important drug target for bone resorption, cancer, and some infectious diseases.…

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Posted in: Bacterial, Cancer Immunology Filed under: Antibacterial, Antitumor, FPPS, UPPS

RPW-24 Possesses Anti-bacterial Activity

2019-11-10 Edward Jenner

Caenorhabditis elegans provides a potential for high throughput, live-animal screening of low molecular weight compound libraries. These are to identify…

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Posted in: Bacterial Filed under: Antibacterial

G907 is a Selective ABC Transporter MsbA Antagonist

2019-10-08 Edward Jenner

ATP binding cassette (ABC) transporters are found in all species. ATP-binding cassette (ABC) transporters constitute a ubiquitous superfamily of integral…

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Posted in: Bacterial Filed under: ABC, Antibacterial, MsbA

MAC13772 is an Inhibitor of the Enzyme BioA with Anti-Bacterial Activity

2019-10-04 Edward Jenner

The alarming spread of multidrug resistance is due to a very limited number of pathways for existing antibiotics. Biotin biosynthesis…

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Posted in: Bacterial Filed under: Antibacterial, BioA

VXc-​486, a Gyrase B Inhibitor, Has Potential to Treat Tuberculosis

2019-09-19 Edward Jenner

Tuberculosis (TB) is an important infectious disease threat worldwide. HIV coinfection/immunosuppression and widespread drug resistance contributes to the challenge of…

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Posted in: Bacterial, Tuberculosis Filed under: Antibacterial, Gyrase, Multidrug Resistance

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