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Tag: Antibacterial

Sulfaphenazole is a Specific CYP2C9 Inhibitor with Antibacterial and Antimicrobial Activity

2022-05-21 Edward Jenner

CYP2C9 is an enzyme protein. The enzyme participates in the metabolism of exogenous substances (including drugs) and endogenous compounds (including…

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Posted in: Bacterial, Inflammation Filed under: Antibacterial, CYP2C9

Xanthoangelol Possesses Antibacterial and Anticancer Activity

2022-04-23 Edward Jenner

Antibacterials usually refer to antibiotics. Specifically, the development of antibiotic-resistant bacteria stems from many factors. Besides, they include the widespread…

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Posted in: Bacterial, Cancer Immunology Filed under: Antibacterial, Anticancer

Ibezapolstat is a First-in-class and Orally Active DNA polymerase IIIC Inhibitor

2021-03-03 Edward Jenner

The Gram-positive obligate anaerobic spore-forming bacterium Clostridioides difficile is a nosocomial pathogen. The severity and prevalence of C. difficile infection (CDI) have caused the…

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Posted in: Infection Filed under: Antibacterial, Anticlostridial, DNA Polymerase

BPH-1358 is a Dual FPPS and UPPS Inhibitor

2019-11-11 Edward Jenner

As we all know, Farnesyl diphosphate synthase(FPPS) is an important drug target for bone resorption, cancer, and some infectious diseases.…

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Posted in: Bacterial, Cancer Immunology Filed under: Antibacterial, Antitumor, FPPS, UPPS

RPW-24 Possesses Anti-bacterial Activity

2019-11-10 Edward Jenner

Caenorhabditis elegans provides a potential for high throughput, live-animal screening of low molecular weight compound libraries. These are to identify…

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Posted in: Bacterial Filed under: Antibacterial

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