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Tag: TLR

Enpatoran is an Orally Active and Dual TLR7/8 Inhibitor

2021-02-27 Edward Jenner

Toll-like receptors 7 and 8 (TLR7/8) are receptors for single-stranded RNA that reside in the endosome. TLR8 mainly expresses in…

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Posted in: Autoimmune Disorders, Systemic Lupus Erythematosus Filed under: Cytokine, IFN-α, IL-6, TLR

MSC2360844 is an Orally Active and Selective PI3Kδ Inhibitor

2020-11-07 Edward Jenner

SLE is a complex autoimmune inflammatory disease that affects multiple organs with unpredictable flares. Autoantibody/antigen immune-complexes in turn can activate…

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Posted in: Autoimmune Disorders, Lupus Nephritis Filed under: IFNα, PI3K, SLE, TLR

3M-011, a Cytokine Inducer, is a Dual TLR7/8 Agonist

2020-05-09 Edward Jenner

3M-011 is a potent dual toll-like receptor TLR7/8 agonist and a cytokine inducer. Firstly, in B16-F10 melanoma cells, 3M-011 treatment can decrease…

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Posted in: Influenza Virus, Viral Immunology Filed under: Cytokine, Melanoma, TLR

CU-T12-9 is a Specific TLR1/2 Agonist

2020-01-01 Edward Jenner

Toll-like receptors belong to a family of pattern recognition receptors, regulate innate immunity and subsequent adaptive immune responses. TLRs can…

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Posted in: Inflammation Filed under: iNOS, Interleukin, TLR, TNF

PF-4878691 is a Selective TLR7 Agonist with HCV Antiviral Efficacy

2019-11-03 Edward Jenner

Chronic hepatitis C (CHC) virus infection continues to be a significant health burden, and 2–3% of the global population infected…

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Posted in: HCV, Inflammation Filed under: Antiviral, HCV, TLR

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  • Enpatoran is an Orally Active and Dual TLR7/8 Inhibitor 2021-02-27
  • WEHI-9625, a VDAC2:BAK Interaction Enhancer, Blocks mBAK-Mediated Apoptosis 2021-02-25
  • S 38093 is a Brain-Penetrant and Orally Active Antagonist of H3 Receptor 2021-02-24

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